(R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Chemical Properties |
Melting point | 116-120°C |
storage temp. | 2-8°C |
solubility | DMSO: soluble20mg/mL |
form | solid |
color | white to off-white |
InChIKey | RATSWNOMCHFQGJ-XODSYJLDSA-N |
CAS DataBase Reference | 183814-30-4 |
Safety Information |
RIDADR | UN 2811 6.1 / PGII |
WGK Germany | 3 |
HS Code | 29242990 |
(R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Usage And Synthesis |
Chemical Properties | Pale Yellow Solid |
Uses | ForMoter ol FuMarate Dihydrate is a selective β2-adrenergic receptor agonist,it is used as an antiasthmatic. |
Uses | A selective β2-adrenergic receptor agonist. Used as an antiasthmatic. |
Biological Activity | Potent, selective and long-acting β 2 -adrenoceptor agonist. Displays 330-fold selectivity for β 2 over β 1 receptors (pK d values are 8.12 and 5.58 respectively). Potently relaxes guinea pig trachea (pD 2 = 9.29), and is longer-acting and 100-fold more potent than salbutam ol. |